Abemaciclib
阿贝西利
Application
Abemaciclib
CAS No. 1231929-97-7
C₂₇H₃₂F₂N₈
Therapeutic Area
52 intermediates
Area Overview
Our oncology portfolio follows the terminal APIs represented in the catalog, spanning kinase inhibitors, DNA-damage and cell-cycle programs, endocrine oncology, and building blocks for ADC and PROTAC development.
Classification is based on terminal APIs in the product catalog; product counts update with the catalog.
Representative Terminal APIs
52 catalog intermediates
阿贝西利
Application
Abemaciclib
CAS No. 1231929-97-7
C₂₇H₃₂F₂N₈
阿达格拉西布
Application
Adagrasib
CAS No. 2326521-71-3
C₃₂H₃₅ClFN₇O₂
(3-氨基-1,2,4-三嗪-6-基)-2-氟苯甲腈
Application
Capmatinib
CAS No. 1197377-47-1
C₁₀H₆FN₅
8-氰基-3-氟苯硼酸频哪酯
Application
Capmatinib
CAS No. 870238-67-8
C₁₃H₁₅BFNO₂
3-氨基-6-溴-1,2,4-三嗪
Application
Capmatinib
CAS No. 69249-22-5
C₃H₃BrN₄
[2-氯-1-羟基-3-(6-喹啉基)丙基]-2,5-吡咯烷二酮
Application
Capmatinib
CAS No. 1197377-31-3
C₁₆H₁₅ClN₂O₃
洛拉替尼
Application
Lorlatinib
CAS No. 1454846-35-5
C₂₁H₁₉FN₆O₂
(S)-叔丁基3-(4-氨基苯基)哌啶-1-甲酸酯
Application
Niraparib
CAS No. 1171197-20-8
C₁₆H₂₄N₂O₂
3-甲酰基-2-硝基苯甲酸甲酯
Application
Niraparib
CAS No. 138229-59-1
C₉H₇NO₅
叔丁基3-(4-氨基苯基)哌啶-1-甲酸酯
Application
Niraparib
CAS No. 875798-79-1
C₁₆H₂₄N₂O₂
奥希替尼
Application
Osimertinib
CAS No. 1421373-65-0
C₂₈H₃₃N₇O₂
2-氯-8-环戊基-5-甲基吡啶并[2,3-d]嘧啶-7(8H)-酮
Application
Palbociclib
CAS No. 1013916-37-4
C₁₃H₁₄ClN₃O
叔丁基4-(6-氨基吡啶-3-基)哌嗪-1-甲酸酯
Application
Palbociclib
CAS No. 571188-59-5
C₁₄H₂₂N₄O₂
瑞博西利
Application
Ribociclib
CAS No. 1211441-98-3
C₂₃H₃₀N₈O
索托拉西布
Application
Sotorasib
CAS No. 2296729-00-3
C₃₀H₃₀F₂N₆O₃
1-甲基-4-(6-氨基吡啶-3-基)哌嗪
Application
Trilaciclib
CAS No. 571189-49-6
C₁₀H₁₆N₄
5-溴-2,4-二氯嘧啶
Application
Trilaciclib
CAS No. 36082-50-5
C₄HBrCl₂N₂
螺[环己烷-1,9'(6'H)-吡嗪并[1',2':1,5]吡咯并[2,3-d]嘧啶]-6'-酮, 2'-氯-7',8'-二氢-
Application
Trilaciclib
CAS No. 1374635-90-1
C₁₄H₁₅ClN₄O
(S)-3-(4-氯苯基)-β-丙氨醇
Application
Capivasertib
CAS No. 886061-26-3
C₉H₁₂ClNO
N-BOC-氨基-哌啶基-1,1-羧酸
Application
Capivasertib
CAS No. 252720-31-3
C₁₁H₂₀N₂O₄
1-(3-氟丙基)氮杂环丁烷-3-胺双(4-甲基苯磺酸盐)
Application
Camizestrant
CAS No. 2231673-65-5
C₂₀H₂₉FN₂O₆S₂
((2R)-1-(1-(1-(四氢-2H-吡喃-2-基)-1H-吲唑-4-基)丙-2-基)氨基甲酸叔丁酯
Application
Camizestrant
CAS No. 2222846-04-8
C₂₀H₂₉N₃O₃
((S)-2-(2-吗啉乙酰胺基)-4-苯基丁酰基)-L-亮氨酰-L-苯丙氨酸
Application
carfilzomib
CAS No. 1690223-94-9
(αS)-α-[[2-(4-吗啉基)乙酰基]氨基]苯丁酰基-L-亮氨酰基-L-苯丙氨酸甲酯
Application
carfilzomib
CAS No. 1140908-89-9
C₃₂H₄₄N₄O₆
2,4,6-三甲基苯磺酰氯
Application
Selpercatinib
CAS No. 773-64-8
C₉H₁₁ClO₂S
4-(6-氟吡啶-3-基)-6-(2-羟基-2-甲基丙氧基)吡唑并[1,5-A]吡啶-3-腈
Application
Selpercatinib
CAS No. 2222653-74-7
C₁₇H₁₅FN₄O₂
6-羟基-4-(6-氟-3-吡啶)-吡唑并[1,5-A]吡啶-3-甲腈
Application
Selpercatinib
CAS No. 2222654-09-1
C₁₃H₇FN₄O
6-(叔丁氧羰基)-3,6-二氮杂双环[3.1.1]庚烷
Application
Selpercatinib
CAS No. 869494-16-6
C₁₀H₁₈N₂O₂
6-甲氧基-3-吡啶甲醛
Application
Selpercatinib
CAS No. 65873-72-5
C₇H₇NO₂
6-溴-4-甲氧基吡唑并[1,5-A]吡啶-3-甲腈
Application
Selpercatinib
CAS No. 1207836-10-9
C₉H₆BrN₃O
N-羟基氨基甲酸叔丁酯; N-叔丁氧羰基羟胺
Application
Selpercatinib
CAS No. 36016-38-3
C₅H₁₁NO₃
1-(1-(3-甲氧基-4-硝基苯基)哌啶-4-基)-4-甲基哌嗪
Application
Brigatinib
CAS No. 761440-65-7
C₁₇H₂₆N₄O₃
2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯胺
Application
Brigatinib
CAS No. 761440-75-9
C₁₇H₂₈N₄O
2,5-二氯-N-[2-(二甲基亚膦酰)苯基]-4-嘧啶胺
Application
Brigatinib
CAS No. 1197953-49-3
C₁₂H₁₂Cl₂N₃OP
(S)-1-氨基丙烷-2-基氨基碳酸甲酯盐酸盐
Application
Encorafenib
CAS No. 1229025-32-4
C₅H₁₃ClN₂O₂
N-[5-氯-2-氟-3-(4,4,5,5-四甲基-1,3,2-二氧杂硼硼烷-2-基)苯基]氨基甲酸叔丁酯
Application
Encorafenib
CAS No. 1269440-69-8
C₁₇H₂₄BClFNO₄
(R)-6-(2-(乙氨基)-4-甲氧基苯基)-5,6,7,8-四氢萘-2-醇
Application
Elacestrant
CAS No. 3033111-52-0
C₁₉H₂₃NO₂
7-苄氧基-3-溴-1,2-二氢萘
Application
Elacestrant
CAS No. 722536-73-4
C₁₇H₁₅BrO
{2-[6-(苄基氧基)-3,4-二氢萘-2-基]-5-甲氧基苯基}(乙基)胺
Application
Elacestrant
CAS No. 3057421-86-7
MC-缬氨酸-瓜氨酸-PABC连接子
Application
ADC Linker
CAS No. 159857-80-4
C₂₈H₄₀N₆O₇
SMCC
Application
ADC Linker
CAS No. 64987-85-5
C₁₆H₁₈N₂O₆
甲磺酸依沙替康
Application
ADC Payload
CAS No. 197720-53-9
C₂₅H₃₀FN₃O₉S
依沙替康衍生物 (DXd)
Application
ADC Payload
CAS No. 1599440-33-1
C₂₆H₂₄FN₃O₆
单甲基奥瑞他汀E (MMAE)
Application
ADC Payload
CAS No. 474645-27-7
C₃₉H₆₇N₅O₇
单甲基奥瑞他汀F (MMAF)
Application
ADC Payload
CAS No. 745017-94-1
C₃₉H₆₅N₅O₈
PBD二聚体 (SG3199)
Application
ADC Payload
CAS No. 1594094-64-0
C₂₃H₂₁IN₂O₃
SN-38
Application
ADC Payload
CAS No. 86639-52-3
C₂₂H₂₀N₂O₅
沙利度胺-NH-PEG4-COOH
Application
PROTAC Linker
CAS No. 1835736-39-4
VH032-PEG4-COOH
Application
PROTAC Linker
CAS No. 2098836-45-2
C₄₈H₅₈ClN₉O₅S₃
4-(4-甲基-1-哌嗪基)-2-[(4-四氢吡喃基)(2,2,2-三氟乙酰基)氨基]苯甲酸三氟乙酸盐
Application
Entrectinib
CAS No. 1034975-62-6
C₂₁H₂₅F₆N₃O₆
5-(3,5-二氟苄基)-1H-吲唑-3-胺
Application
Entrectinib
CAS No. 1108745-30-7
C₁₄H₁₁F₂N₃
5-(3,5-二氟苄基)-2-氟苄腈;2-氟-5-(3,5-二氟苄基)苯腈
Application
Entrectinib
CAS No. 1108745-25-0
C₁₄H₈F₃N
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